SCHEMBL3363192

SCHEMBL3363192

COc1cc2c(CC(=O)N(C)Cc3cccnc3)cnc(CNC(=O)OC(C)(C)C)c2cc1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.41
RECQL P46063 1/20 0.41
ALDH1A1 P00352 6/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
USP2 O75604 1/20 0.40
NAMPT P43490 1/20 0.40
RIPK1 Q13546 1/20 0.39
HPGD P15428 3/20 0.38
DPP4 P27487 2/20 0.38
HSD17B10 Q99714 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPK1 P28482 1/20 0.38
PDE10A Q9Y233 1/20 0.38
PKM P14618 2/20 0.38
ALOX12 P18054 1/20 0.38
CYP1A2 P05177 2/20 0.38
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3361800 0.92 CTSL (0.43) L3MBTL1DPP4MAPK1MAPTMEN1
SCHEMBL3363215 0.83 DPP4 (0.56) RECQLALDH1A1RIPK1HPGDDPP4
Hydrochloric Acid SCHEMBL3361965 0.83 DPP4 (0.57) RECQLALDH1A1RIPK1HPGDDPP4
SCHEMBL3360434 0.82 DPP4 (0.41) ALDH1A1DPP4PDE10AMEN1KMT2A
SCHEMBL3365064 0.81 KDM4E (0.43) ALDH1A1NPSR1DPP4KDM4EPDE10A
SCHEMBL3363185 0.79 NAMPT (0.39) CYP3A4RECQLALDH1A1L3MBTL1NPSR1
SCHEMBL3362959 0.79 DPP4 (0.40) DPP4PDE10A
SCHEMBL3361880 0.78 DPP4 (0.47) DPP4PDE10A
SCHEMBL3362196 0.78 DPP4 (0.46) DPP4PDE10A
SCHEMBL3361175 0.78 HPGD (0.44) HPGDDPP4MAPTHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed