SCHEMBL3365202

SCHEMBL3365202

COc1ccc(CNC(=O)c2cnc(CNC(=O)OC(C)(C)C)c3c(OC)cc(OC)cc23)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
RAB9A P51151 1/20 0.44
CYP1A2 P05177 1/20 0.44
POLB P06746 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ATM Q13315 1/20 0.44
MAPT P10636 3/20 0.43
KDM4E B2RXH2 3/20 0.43
PKM P14618 1/20 0.43
LMNA P02545 2/20 0.43
PDE10A Q9Y233 1/20 0.42
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
TP53 P04637 1/20 0.42
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3365143 0.88 PDE10A (0.51) DPP4ALDH1A1HPGDL3MBTL1RAB9A
SCHEMBL3361298 0.87 DPP4 (0.46) DPP4ALDH1A1HPGDRAB9ACYP1A2
SCHEMBL3363099 0.86 DPP4 (0.49) DPP4ALDH1A1L3MBTL1CYP1A2LMNA
SCHEMBL3362414 0.85 DPP4 (0.61) DPP4ALDH1A1HPGDL3MBTL1RAB9A
Hydrochloric Acid SCHEMBL3361903 0.84 DPP4 (0.62) DPP4ALDH1A1HPGDL3MBTL1RAB9A
SCHEMBL3362101 0.82 DPP4 (0.67) DPP4ALDH1A1HPGDRAB9AMAPT
SCHEMBL3362437 0.81 DPP4 (0.45) DPP4ALDH1A1L3MBTL1TSHRHSD17B10
SCHEMBL3365615 0.80 DPP4 (0.41) DPP4ALDH1A1HPGDL3MBTL1KDM4E
SCHEMBL3361307 0.80 DPP4 (0.46) DPP4ALDH1A1L3MBTL1MAPTLMNA
SCHEMBL3359830 0.79 NAMPT (0.44) DPP4ALDH1A1HPGDL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed