SCHEMBL3367655

SCHEMBL3367655

O=C(O)Cn1cc2cccc(-c3ccc(Cl)cc3Cl)c2n1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MARS1 P56192 3/20 0.44
CRHR1 P34998 5/20 0.42
CNR1 P21554 6/20 0.42
PARP1 P09874 1/20 0.40
CNR2 P34972 1/20 0.38
KMO O15229 1/20 0.38
SHMT1 P34896 1/20 0.37
SHMT2 P34897 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3364716 0.84 CNR1 (0.46) CRHR1CNR1
SCHEMBL3364790 0.82 PARP1 (0.50) MARS1CRHR1CNR1PARP1
SCHEMBL3364024 0.82 CRHR1 (0.49) CRHR1
Trifluoroacetic Acid SCHEMBL3364681 0.81 PARP1 (0.50) MARS1CRHR1CNR1PARP1
SCHEMBL3361832 0.75 CRHR1 (0.52) CRHR1
Hydrochloric Acid SCHEMBL3364528 0.74 CRHR1 (0.51) CRHR1
SCHEMBL23320986 0.72 EPHX2 (0.47) PARP1
SCHEMBL12985765 0.72 PARP1 (0.45) PARP1
SCHEMBL4662108 0.68 CRHR1 (0.50) CRHR1
SCHEMBL3363050 0.67 MARS1 (0.50) MARS1CRHR1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656353-B1 GABANERGIC MODULATORS HOFFMANN LA ROCHE (CH) 2010-01-27 EP claimed