SCHEMBL3368095

SCHEMBL3368095

O=C(O)c1ccc(C(O)(c2ccccc2)c2ccccc2Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.52
CYP3A5 P20815 1/20 0.52
CYP19A1 P11511 1/20 0.51
KCNN4 O15554 1/20 0.44
TSHR P16473 4/20 0.42
ALOX15 P16050 1/20 0.42
DAO P14920 1/20 0.42
NAPRT Q6XQN6 1/20 0.42
HPGD P15428 1/20 0.42
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
NR4A2 P43354 1/20 0.42
SRD5A2 P31213 4/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRK1 P41145 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2131459 0.86 CYP3A4 (0.60) CYP3A4CYP3A5CYP19A1KCNN4TSHR
SCHEMBL30114522 0.86 CYP3A4 (0.60) CYP3A4CYP3A5CYP19A1KCNN4TSHR
SCHEMBL34463323 0.84 CYP3A4 (0.48) CYP3A4CYP3A5CYP19A1KCNN4TSHR
SCHEMBL675338 0.82 CYP3A4 (0.71) CYP3A4CYP3A5CYP19A1KCNN4TSHR
SCHEMBL407595 0.82 TSHR (0.56) TSHRALOX15DAONAPRTRXRA
SCHEMBL6369689 0.82 KCNN4 (0.57) CYP3A4CYP3A5CYP19A1KCNN4TSHR
SCHEMBL4466320 0.81 CYP3A4 (0.56) CYP3A4CYP3A5CYP19A1KCNN4TSHR
SCHEMBL14156831 0.79 CYP3A4 (0.55) CYP3A4CYP3A5CYP19A1KCNN4HTR2A
SCHEMBL6558548 0.75 SLC2A1 (0.56) CYP3A4CYP3A5CYP19A1KCNN4TSHR
SCHEMBL4460626 0.75 CYP3A4 (0.51) CYP3A4CYP3A5CYP19A1KCNN4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2159228-A1 Amphiphilic solid support Polymer Laboratories Limited (GB) 2010-03-03 EP disclosed