SCHEMBL3368239

SCHEMBL3368239

O=C(O)ON1CCCC1c1nnc(-c2cccnc2)o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
MAPK1 P28482 2/20 0.45
GAA P10253 1/20 0.44
HCRTR1 O43613 4/20 0.44
HCRTR2 O43614 4/20 0.44
TNKS O95271 2/20 0.44
PARP1 P09874 2/20 0.44
PARP2 Q9UGN5 2/20 0.44
USP30 Q70CQ3 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
KCNH2 Q12809 1/20 0.42
SCD O00767 1/20 0.42
RAB9A P51151 2/20 0.41
EGFR P00533 1/20 0.41
PTGS2 P35354 1/20 0.41
CYP1A2 P05177 2/20 0.40
MAPT P10636 1/20 0.40
GPR55 Q9Y2T6 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3370373 0.89 USP30 (0.51) ALDH1A1MAPK1HCRTR1HCRTR2TNKS
SCHEMBL3366782 0.87 USP30 (0.52) ALDH1A1MAPK1HCRTR1HCRTR2USP30
SCHEMBL3368236 0.84 ALDH1A1 (0.56) ALDH1A1MAPK1GAAHCRTR1HCRTR2
SCHEMBL3368153 0.81 HCRTR1 (0.58) ALDH1A1MAPK1GAAHCRTR1HCRTR2
SCHEMBL3366568 0.80 ALDH1A1 (0.54) ALDH1A1HCRTR1HCRTR2
SCHEMBL3369474 0.77 HCRTR1 (0.47) HCRTR1HCRTR2TNKSPARP1PARP2
SCHEMBL3370346 0.76 HCRTR2 (0.52) ALDH1A1HCRTR1HCRTR2SCDRAB9A
SCHEMBL3370671 0.76 HCRTR2 (0.49) ALDH1A1HCRTR1HCRTR2KCNH2SCD
SCHEMBL3370256 0.76 HCRTR2 (0.49) ALDH1A1HCRTR1HCRTR2KCNH2SCD
SCHEMBL3366725 0.75 ALDH1A1 (0.51) ALDH1A1GAAHCRTR1HCRTR2TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532141-B1 2-PYRROLIDIN-2-YL- [1,3,4]-OXADIAZOLE DERIVATIVES AND THE USE OF THE SAME AS ANTIDEPRESSANTS GRUENENTHAL GMBH (DE) 2010-10-13 EP disclosed