SCHEMBL3368784

SCHEMBL3368784

COc1cc(-c2cc(-c3cncc(C(=O)NC(C)CO)c3)cn2S(=O)(=O)c2cc(O)ccc2C)cc(OC)c1OC

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.36
MAPK1 P28482 1/20 0.36
CTSA P10619 4/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
XDH P47989 5/20 0.34
ACVR1 Q04771 2/20 0.33
APLNR P35414 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TGFBR1 P36897 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1379796 0.86 MAPK1 (0.38) SYKMAPK1CTSAXDHACVR1
SCHEMBL3369860 0.85 L3MBTL1 (0.40) NPC1PKMHSD17B10
SCHEMBL3371912 0.82 FYN (0.34) NPC1PKMACVR1TGFBR1
SCHEMBL3370766 0.81 CD274 (0.42) NPC1KDM4EALDH1A1
SCHEMBL3372486 0.80 KDM4E (0.35) NPC1PKMACVR1KDM4EALDH1A1
SCHEMBL3370431 0.76 MAP3K11 (0.45) NPC1PKMTGFBR1
SCHEMBL1376476 0.70 MAP3K11 (0.42) MAPK1PKMACVR1ALDH1A1HSD17B10
SCHEMBL1378956 0.68 CYP11B1 (0.47) PKMALDH1A1
SCHEMBL1376787 0.67 CD274 (0.44) NPC1KDM4EALDH1A1
SCHEMBL3367765 0.67 TUBB4A (0.38) MAPK1NPC1PKMKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1628957-B1 SULFOPYRROLES TAKEDA PHARMACEUTICAL (JP) 2010-09-29 EP claimed