SCHEMBL3370237

SCHEMBL3370237

CCCCCc1ccc2c(c1)NCN2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.43
ADRA2A P08913 2/20 0.43
ADORA3 P0DMS8 2/20 0.43
TACR2 P21452 2/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
SHBG P04278 1/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 1/20 0.43
HSPD1 P10809 1/20 0.43
ADRB3 P13945 1/20 0.43
HTR2C P28335 1/20 0.43
HSPE1 P61604 1/20 0.43
HIF1A Q16665 1/20 0.43
TST Q16762 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16722721 0.89 ESR1 (0.43) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL23519530 0.87 HTR1A (0.43) HTR2CHTR2ASIGMAR1LPLLIPG
SCHEMBL31351356 0.79 PTGS2 (0.52) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL29242122 0.79 PTGS2 (0.52) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL27610237 0.75 DRD2 (0.46) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL27610259 0.75 SMN1; SMN2 (0.44) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL27091898 0.74 SLC6A2 (0.46) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL20846119 0.73 SMN1; SMN2 (0.43) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL565857 0.73 DRD2 (0.45) ESR1ADRA2AADORA3TACR2SLC6A2
SCHEMBL24037195 0.71 PTGS2 (0.47) ESR1ADRA2AADORA3TACR2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9517240-B2 Methods and compositions for cancer prevention and treatment THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-12-13 US disclosed
US-20130331365-A1 METHODS AND COMPOSITIONS FOR CANCER PREVENTION AND TREATMENT THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-12-12 US disclosed
US-20100160275-A1 METHODS AND COMPOSITIONS FOR CANCER PREVENTION AND TREATMENT THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2010-06-24 US disclosed
WO-2008039482-A2 METHODS AND COMPOSITIONS FOR CANCER PREVENTION AND TREATMENT THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2008-04-03 WO disclosed