SCHEMBL3373983

SCHEMBL3373983

O=Cc1ccc2c(=O)[nH]c(=O)[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.56
PARP1 P09874 6/20 0.50
KDM4E B2RXH2 3/20 0.50
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP2A6 P11509 2/20 0.42
TTK P33981 1/20 0.40
GSK3B P49841 2/20 0.36
TYMP P19971 2/20 0.36
BACE1 P56817 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
PTGS2 P35354 1/20 0.35
RAB9A P51151 1/20 0.35
PARG Q86W56 1/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7029179 0.84 PARP1 (0.48) KIF11PARP1KDM4ECA12CA9
SCHEMBL7022549 0.81 PARP1 (0.46) KIF11PARP1KDM4ECA12CA9
SCHEMBL7022550 0.81 PARP1 (0.46) KIF11PARP1KDM4ECA12CA9
SCHEMBL29519732 0.80 KIF11 (0.48) KIF11KDM4EALDH1A1CYP2A6PDE3B
SCHEMBL1418732 0.80 KIF11 (0.48) KIF11KDM4EALDH1A1CYP2A6PDE3B
SCHEMBL28589579 0.80 KIF11 (0.81) KIF11KDM4EALDH1A1CYP2A6TTK
SCHEMBL3380432 0.80 KDM4E (0.53) KIF11PARP1KDM4ECA12CA9
SCHEMBL3380424 0.80 KDM4E (0.53) KIF11PARP1KDM4ECA12CA9
SCHEMBL7033757 0.77 TYMP (0.43) KIF11PARP1KDM4ECA12CA9
SCHEMBL7033759 0.77 TYMP (0.43) KIF11PARP1KDM4ECA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046388-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUINOLIN-2-ONES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed
WO-2010046388-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUINOLIN-2-ONES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed