SCHEMBL3380432

SCHEMBL3380432

O=c1[nH]c(=O)c2ccc(C=Cc3ccccc3)cc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.53
CA12 O43570 1/20 0.53
PARP1 P09874 1/20 0.53
CA9 Q16790 1/20 0.53
IP6K1 Q92551 2/20 0.51
DPYD Q12882 1/20 0.47
KMT2A Q03164 2/20 0.46
IP6K3 Q96PC2 1/20 0.46
IP6K2 Q9UHH9 1/20 0.46
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
TUBB4A P04350 8/20 0.45
TUBB P07437 8/20 0.45
TUBA3C P0DPH7 8/20 0.45
TUBA1B P68363 8/20 0.45
TUBA4A P68366 8/20 0.45
TUBB4B P68371 8/20 0.45
TUBB3 Q13509 8/20 0.45
TUBB2A Q13885 8/20 0.45
TUBB8 Q3ZCM7 8/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3380424 1.00 KDM4E (0.53) KDM4ECA12PARP1CA9IP6K1
SCHEMBL7022550 0.82 PARP1 (0.46) KDM4ECA12PARP1CA9IP6K1
SCHEMBL7022549 0.82 PARP1 (0.46) KDM4ECA12PARP1CA9IP6K1
SCHEMBL3373983 0.80 KIF11 (0.56) KDM4ECA12PARP1CA9RAB9A
SCHEMBL7024202 0.78 PARP1 (0.42) KDM4ECA12PARP1CA9IP6K1
SCHEMBL7024197 0.78 PARP1 (0.42) KDM4ECA12PARP1CA9IP6K1
SCHEMBL7033757 0.78 TYMP (0.43) KDM4ECA12PARP1CA9IP6K1
SCHEMBL7033759 0.78 TYMP (0.43) KDM4ECA12PARP1CA9IP6K1
SCHEMBL7029179 0.78 PARP1 (0.48) KDM4ECA12PARP1CA9DPYD
SCHEMBL7027670 0.76 TYMP (0.46) KDM4ECA12PARP1CA9IP6K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046388-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUINOLIN-2-ONES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed