SCHEMBL3375552

SCHEMBL3375552

NC(=O)C1CN(CCc2ccccc2F)CC1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.40
KCNH2 Q12809 5/20 0.39
TRPM8 Q7Z2W7 1/20 0.38
MC4R P32245 2/20 0.38
SIRT2 Q8IXJ6 2/20 0.38
SIRT1 Q96EB6 2/20 0.38
MCHR1 Q99705 2/20 0.37
SCN3A Q9NY46 5/20 0.37
SCN1A P35498 1/20 0.37
SCN4A P35499 1/20 0.37
SCN7A Q01118 1/20 0.37
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN8A Q9UQD0 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
PRCP P42785 2/20 0.37
TACR1 P25103 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2B6 P20813 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3380618 0.83 PRCP (0.47) CACNA1GMCHR1PRCPTACR1
Hydrochloric Acid SCHEMBL22607752 0.81 SIRT2 (0.46) CACNA1GKCNH2SIRT2SIRT1SCN3A
SCHEMBL3375549 0.74 MC4R (0.39) TRPM8MC4R
Hydrochloric Acid SCHEMBL28626980 0.74 SIRT2 (0.44) KCNH2SIRT2SIRT1MAOB
SCHEMBL3378694 0.71 MCHR1 (0.46) KCNH2MCHR1PRCP
SCHEMBL3345498 0.70 RORC (0.57) KCNH2MC4R
SCHEMBL9556728 0.69 CACNA1G (0.54) CACNA1GMAOB
SCHEMBL3346208 0.69 RORC (0.58) MC4RMCHR1MAOB
SCHEMBL22398100 0.68 FFAR1 (0.53) KCNH2CYP1A2MAOBCYP2C19
SCHEMBL18685562 0.67 NTRK1 (0.51) MC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed