SCHEMBL3375645

SCHEMBL3375645

COC(=O)c1cc(B2OC(C)(C)C(C)(C)O2)cnc1OC1CCN(C)C1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.41
USP30 Q70CQ3 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.36
CHEK1 O14757 3/20 0.36
CHEK2 O96017 1/20 0.36
DGAT1 O75907 1/20 0.35
ALPL P05186 1/20 0.34
KCNH2 Q12809 1/20 0.34
PIK3CD O00329 3/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19499252 0.84 ROCK2 (0.48) ROCK2USP30CHEK2KCNH2
SCHEMBL789862 0.79 ALPL (0.46) ROCK2USP30DGAT1ALPLGSK3A
SCHEMBL29604061 0.79 ALPL (0.46) ROCK2USP30DGAT1ALPLGSK3A
SCHEMBL3342229 0.79 OPRK1 (0.51)
SCHEMBL19499254 0.77 KCNH2 (0.42) ROCK2USP30IRAK4KCNH2
SCHEMBL3345874 0.77 CHEK1 (0.37) CHEK1CHEK2PIK3CDPIK3CAPIK3CB
SCHEMBL25932086 0.76 LRRK2 (0.37) ROCK2USP30ALPLPIK3CD
SCHEMBL16175408 0.76 MALT1 (0.37) ROCK2USP30KCNH2
SCHEMBL3448683 0.75 GAA (0.41) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL19468772 0.75 ROCK2 (0.46) ROCK2USP30DGAT1ALPLKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed