SCHEMBL3375932

SCHEMBL3375932

COC(=O)OCc1cc(-c2cccc(Cl)c2)c2nc(C)c(C3C=CN(C(=O)OC)C=C3)n2c1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 10/20 0.35
ATM Q13315 1/20 0.33
PDE4D Q08499 1/20 0.32
DHODH Q02127 1/20 0.32
EGFR P00533 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRB2 P47870 1/20 0.31
KMT2A Q03164 1/20 0.31
THRB P10828 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7911720 0.90 CHRM3 (0.33) CHRM3ATMPDE4DEGFRGABRA2
SCHEMBL7931506 0.83 PDE4D (0.36) CHRM3ATMPDE4DTHRB
SCHEMBL3378468 0.83 PDE4D (0.38) CHRM3ATMPDE4DEGFRGABRA2
SCHEMBL3379763 0.76 TRPM8 (0.39) CHRM3PDE4DEGFRGABRA2GABRB2
SCHEMBL3381843 0.75 GPR119 (0.39) CHRM3PDE4DEGFRKMT2AHPGD
SCHEMBL7913069 0.73 HDAC6 (0.44) CHRM3PDE4DEGFR
SCHEMBL10442054 0.66 PDE4D (0.47) PDE4DEGFRTHRBNPC1ALDH1A1
SCHEMBL7921942 0.66 CHRM3 (0.31) CHRM3KMT2AALDH1A1
SCHEMBL7916793 0.66 DPP4 (0.39) KMT2ATHRBALDH1A1HPGDSMN1; SMN2
SCHEMBL3466382 0.66 PDE4D (0.62) PDE4DALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO disclosed