SCHEMBL3376187

SCHEMBL3376187

CC(=O)OCC(COC(C)=O)Oc1cccc2c1CCN2

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.35
ADRA2B P18089 2/20 0.35
ADRA2C P18825 2/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
HTR1A P08908 2/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
OPRK1 P41145 1/20 0.33
MTNR1A P48039 2/20 0.32
BRD4 O60885 2/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
PDGFRB P09619 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13337352 0.78 S1PR1 (0.36) MTNR1ABRD4S1PR1S1PR3PDGFRB
SCHEMBL6687227 0.78 MAPK1 (0.41)
SCHEMBL15451257 0.76 KMT2A (0.49)
SCHEMBL15451247 0.75 PPARA (0.41) MTNR1A
SCHEMBL15451286 0.75 PPARA (0.41) MTNR1A
SCHEMBL6687224 0.75 CRBN (0.34) PRMT5WDR77HTR1AMTNR1ABRD4
SCHEMBL3376891 0.75 ADRB2 (0.34) ADRA2AADRA2BADRA2CHTR1AADRB2
SCHEMBL20373858 0.74 NISCH (0.42) ADRA2AADRA2BADRA2CS1PR1S1PR3
SCHEMBL13003057 0.74 ADRA2A (0.33) ADRA2AADRA2BADRA2C
SCHEMBL3304107 0.72 LMNA (0.44) PRMT5WDR77BRD4S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1757585-B1 Anionically substituted 7-Nitroindoline derivatives and their uses MEDICAL RES COUNCIL (GB) 2010-12-01 EP disclosed
US-7737169-B2 Anionically substituted 7-nitroindoline derivatives and their uses MEDICAL RESEARCH COUNCIL (GB) 2010-06-15 US disclosed
EP-1757585-A1 Anionically substituted 7-Nitroindoline derivatives and their uses Medical Research Council (GB) 2007-02-28 EP disclosed