SCHEMBL3377147

SCHEMBL3377147

CS(=O)(=O)N(Cc1ccccc1)c1cccc(C(=O)N2CCCC(c3ccccc3)C2)c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 3/20 0.52
LMNA P02545 2/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PARP14 Q460N5 1/20 0.49
PARP10 Q53GL7 1/20 0.49
ALDH1A1 P00352 5/20 0.49
HPGD P15428 3/20 0.49
TSHR P16473 1/20 0.49
HIF1A Q16665 1/20 0.49
GAA P10253 1/20 0.48
MYC P01106 2/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3377977 0.90 LMNA (0.52) PROKR1LMNAPARP14PARP10ALDH1A1
SCHEMBL302061 0.89 LMNA (0.54) LMNAHTTSMN1; SMN2PARP14PARP10
SCHEMBL3378993 0.83 LMNA (0.48) LMNAHTTSMN1; SMN2ALDH1A1HPGD
SCHEMBL302689 0.80 LMNA (0.37) PROKR1LMNASMN1; SMN2ALDH1A1HPGD
SCHEMBL3377001 0.79 F10 (0.56) LMNAHTTSMN1; SMN2ALDH1A1HPGD
SCHEMBL303313 0.78 LMNA (0.57) LMNAPARP14PARP10ALDH1A1HPGD
SCHEMBL17075498 0.78 LMNA (0.45) LMNAHTTSMN1; SMN2PARP14PARP10
SCHEMBL302677 0.77 F10 (0.47) LMNAHTTSMN1; SMN2ALDH1A1HPGD
SCHEMBL6744201 0.74 KMT2A (0.69) LMNAALDH1A1TSHRGAAMEN1
SCHEMBL304021 0.73 PROKR1 (0.49) PROKR1LMNAHTTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9073834-B2 Potassium channel blockers XENTION LIMITED (GB) 2015-07-07 US claimed
US-20140221337-A1 Potassium Channel Blockers XENTION LIMITED (GB) 2014-08-07 US claimed
US-20100087428-A1 Novel Potassium Channel Blockers XENTION LIMITED (GB) 2010-04-08 US claimed
EP-2342177-B1 NOVEL POTASSIUM CHANNEL BLOCKERS JAPAN TOBACCO INC (JP) 2017-02-15 EP disclosed
US-9073834-B2 Potassium channel blockers XENTION LIMITED (GB) 2015-07-07 US disclosed
US-20140221337-A1 Potassium Channel Blockers XENTION LIMITED (GB) 2014-08-07 US disclosed
US-8673901-B2 Potassium channel blockers XENTION LIMITED (GB) 2014-03-18 US disclosed
US-20100087428-A1 Novel Potassium Channel Blockers XENTION LIMITED (GB) 2010-04-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221337-A1 Potassium Channel Blockers KCNJ2, KCNH2, KCNB1 PROKR1 1828/4885LMNA 1619/4885HTT 2305/4885
US-20100087428-A1 Novel Potassium Channel Blockers HCN4, SCN2B, KCNH2 PROKR1 817/4885LMNA 2145/4885HTT 2035/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.