SCHEMBL3377517

SCHEMBL3377517

CCOC(=O)Oc1cncc2ccsc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.36
MAPT P10636 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
PKM P14618 2/20 0.35
POLB P06746 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
ALDH1A1 P00352 3/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CA2 P00918 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
KDM4E B2RXH2 2/20 0.34
CYP3A4 P08684 1/20 0.34
GAA P10253 1/20 0.34
CUL4A Q13619 2/20 0.34
TYMS P04818 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28949857 0.82 KDM4E (0.39) MAPTRAB9APOLBALDH1A1KMT2A
SCHEMBL27739264 0.77 TSHR (0.45) MAPTNPC1RAB9APKMPOLB
SCHEMBL8516383 0.69 TSHR (0.52) ALOX5MAPTPOLBALDH1A1KMT2A
SCHEMBL19020580 0.69 PDE10A (0.36)
SCHEMBL3842038 0.68 GABRA1 (0.39) MAPTALDH1A1KMT2AMEN1CYP1A2
SCHEMBL29480246 0.68 MEN1 (0.41) POLBALDH1A1KMT2AMEN1CA2
SCHEMBL7456124 0.66 ALDH1A1 (0.51) MAPTNPC1RAB9APKMNPSR1
SCHEMBL1958548 0.66 TYMS (0.49) ALOX5MAPTNPC1RAB9APOLB
SCHEMBL11727074 0.66 CYP2A6 (0.42) CYP2C9CYP2C19CYP3A4ICAM1SELE
SCHEMBL7785899 0.66 ALDH1A1 (0.38) ALOX5ALDH1A1KMT2ACA2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038288-B1 NOVEL 4-AMINO-3-(-AZOLYL-PHENOXYMETHYL)-THIENOÝ3,2¨PYRIDINE-7-CARBOXYLIC ACID DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-11-24 EP claimed