SCHEMBL3377895

SCHEMBL3377895

N#Cc1cccc(N)c1-c1ncccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CLK4 Q9HAZ1 1/20 0.41
HDAC1 Q13547 1/20 0.40
ALDH1A1 P00352 4/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
MAP2K1 Q02750 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
KDM4E B2RXH2 2/20 0.37
HTT P42858 1/20 0.36
CYP19A1 P11511 1/20 0.36
HPGD P15428 2/20 0.36
CYP2D6 P10635 1/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21899485 0.82 CYP3A4 (0.50) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL2732615 0.81 TSHR (0.50) CYP1A2CYP3A4CYP2C9CYP2C19CLK4
SCHEMBL22232393 0.80 ADRB2 (0.41) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL1586204 0.78 CLK4 (0.41) CYP1A2CYP3A4CYP2C9CYP2C19CLK4
SCHEMBL29912400 0.78 CLK4 (0.41) CYP1A2CYP3A4CYP2C9CYP2C19CLK4
SCHEMBL11963779 0.76 GRM5 (0.48) CYP1A2CYP3A4CYP2C9CYP2C19MAP2K1
SCHEMBL1848389 0.75 PDPK1 (0.40) CYP1A2CYP3A4CYP2C9CYP2C19HDAC1
SCHEMBL3377900 0.74 CLK4 (0.41) CYP1A2CYP3A4CYP2C9CYP2C19CLK4
SCHEMBL27510138 0.73 CYP1A2 (0.47) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL3259923 0.73 CYP1A2 (0.47) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9427400-B2 Platinum-catalyzed intravaginal rings INTERNATIONAL PARTNERSHIP FOR MICROBICIDES (US) 2016-08-30 US disclosed
US-20140056961-A1 PLATINUM-CATALYZED INTRAVAGINAL RINGS INTERNATIONAL PARTNERSHIP FOR MICROBICIDES (US) 2014-02-27 US disclosed
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140056961-A1 PLATINUM-CATALYZED INTRAVAGINAL RINGS PCNA, DPYD, QDPR CYP1A2 719/4885CYP3A4 287/4885CYP2C9 568/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.