SCHEMBL3378593

SCHEMBL3378593

Cn1c(=O)ccc2ncc(C#N)c(OCC3CCC(N)CC3)c21

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.39
ABL1 P00519 7/20 0.36
SRC P12931 7/20 0.36
ABL2 P42684 7/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
XDH P47989 1/20 0.35
KDM1A O60341 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
KCNH2 Q12809 1/20 0.34
SSTR2 P30874 1/20 0.33
LRRK2 Q5S007 1/20 0.33
PRKCQ Q04759 1/20 0.33
MELK Q14680 1/20 0.33
DPP4 P27487 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3378590 1.00 CHEK1 (0.39) CHEK1ABL1SRCABL2TLR9
SCHEMBL3375050 0.86 TLR9 (0.40) CHEK1TLR9TLR8TLR7KDM1A
SCHEMBL3379792 0.86 RORC (0.38) CHEK1ABL1SRCABL2TLR9
SCHEMBL3379795 0.86 RORC (0.38) CHEK1ABL1SRCABL2TLR9
SCHEMBL3375046 0.86 TLR9 (0.40) CHEK1TLR9TLR8TLR7KDM1A
Hydrochloric Acid SCHEMBL3377052 0.85 TLR9 (0.39) CHEK1TLR9TLR8TLR7KDM1A
Hydrochloric Acid SCHEMBL3377057 0.85 TLR9 (0.39) CHEK1TLR9TLR8TLR7KDM1A
SCHEMBL3352394 0.84 KCNH2 (0.41) ABL1SRCABL2XDHKCNH2
SCHEMBL3352400 0.84 KCNH2 (0.41) ABL1SRCABL2XDHKCNH2
SCHEMBL3378582 0.81 RORC (0.33) ABL1SRCABL2XDHKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046388-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUINOLIN-2-ONES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed