SCHEMBL3352400

SCHEMBL3352400

Cn1c(=O)ccc2ncc(C#N)c(OCC3CCC(NC(=O)O)CC3)c21

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.41
XDH P47989 2/20 0.36
SSTR4 P31391 3/20 0.36
ABL1 P00519 4/20 0.35
SRC P12931 4/20 0.35
ABL2 P42684 4/20 0.35
PDE4B Q07343 1/20 0.35
PDE4D Q08499 1/20 0.35
RORC P51449 1/20 0.35
LRRK2 Q5S007 1/20 0.34
KCNJ1 P48048 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3352394 1.00 KCNH2 (0.41) KCNH2XDHSSTR4ABL1SRC
SCHEMBL3345358 0.87 LRRK2 (0.41) KCNH2SSTR4RORCLRRK2
SCHEMBL3347090 0.87 RORC (0.40) KCNH2PDE4DRORC
SCHEMBL3345353 0.87 LRRK2 (0.41) KCNH2SSTR4RORCLRRK2
SCHEMBL3347085 0.87 RORC (0.40) KCNH2PDE4DRORC
SCHEMBL3378590 0.84 CHEK1 (0.39) KCNH2XDHABL1SRCABL2
SCHEMBL3378593 0.84 CHEK1 (0.39) KCNH2XDHABL1SRCABL2
SCHEMBL3345752 0.83 LRRK2 (0.39) RORCLRRK2
SCHEMBL3345749 0.83 LRRK2 (0.39) RORCLRRK2
SCHEMBL3345692 0.82 LRRK2 (0.37) KCNH2SSTR4LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045987-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUIN0LIN-2-0NES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed