SCHEMBL3379792

SCHEMBL3379792

Cn1c(=O)ccc2ncc(Cl)c(OC[C@H]3CC[C@H](N)CC3)c21

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.38
PDE4D Q08499 1/20 0.37
CHEK1 O14757 1/20 0.35
CNR2 P34972 2/20 0.34
TLR9 Q9NR96 1/20 0.34
TLR8 Q9NR97 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
MELK Q14680 2/20 0.34
LRRK2 Q5S007 1/20 0.34
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
GRM2 Q14416 4/20 0.33
ABL1 P00519 1/20 0.33
SRC P12931 1/20 0.33
ABL2 P42684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3379795 1.00 RORC (0.38) RORCPDE4DCHEK1CNR2TLR9
SCHEMBL3375050 0.87 TLR9 (0.40) RORCCHEK1TLR9TLR8TLR7
SCHEMBL3375046 0.87 TLR9 (0.40) RORCCHEK1TLR9TLR8TLR7
SCHEMBL3378590 0.86 CHEK1 (0.39) CHEK1TLR9TLR8TLR7MELK
SCHEMBL3378593 0.86 CHEK1 (0.39) CHEK1TLR9TLR8TLR7MELK
Hydrochloric Acid SCHEMBL3377057 0.86 TLR9 (0.39) RORCCHEK1TLR9TLR8TLR7
Hydrochloric Acid SCHEMBL3377052 0.86 TLR9 (0.39) RORCCHEK1TLR9TLR8TLR7
SCHEMBL3347085 0.83 RORC (0.40) RORCPDE4DCNR2
SCHEMBL3347090 0.83 RORC (0.40) RORCPDE4DCNR2
SCHEMBL3352142 0.80 RORC (0.38) RORCPDE4DCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045987-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUIN0LIN-2-0NES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed