SCHEMBL3378982

SCHEMBL3378982

O=C(NCC1CC(Oc2cccc(CN3CCCC3)c2Cl)C1)OC1CCOCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.40
CYP2A13 Q16696 1/20 0.38
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
CXCR4 P61073 1/20 0.36
GSK3B P49841 1/20 0.36
KCNH2 Q12809 1/20 0.36
ACACB O00763 1/20 0.36
ACACA Q13085 1/20 0.36
TP53 P04637 2/20 0.35
ALPL P05186 1/20 0.35
ALPI P09923 1/20 0.35
ALPG P10696 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
BCHE P06276 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3378894 0.87 P2RX7 (0.43) P2RX7KDM4EALDH1A1POLBCXCR4
SCHEMBL3380633 0.82 P2RX7 (0.41) P2RX7KDM4EALDH1A1POLBCXCR4
SCHEMBL3377159 0.82 HRH3 (0.41) P2RX7CYP2A13KDM4EALDH1A1POLB
SCHEMBL4646894 0.80 P2RX7 (0.41) P2RX7KDM4EALDH1A1POLBTP53
SCHEMBL4647815 0.80 P2RX7 (0.43) P2RX7KDM4EALDH1A1POLBCXCR4
SCHEMBL3378700 0.79 P2RX7 (0.37) P2RX7KDM4EALDH1A1POLBCXCR4
SCHEMBL4648735 0.79 P2RX7 (0.39) P2RX7KDM4EALDH1A1POLBCXCR4
Hydrochloric Acid SCHEMBL3379328 0.79 P2RX7 (0.44) P2RX7KDM4EALDH1A1POLBCXCR4
Hydrochloric Acid SCHEMBL3379330 0.79 P2RX7 (0.44) P2RX7KDM4EALDH1A1POLBCXCR4
SCHEMBL3376438 0.78 CYP2A13 (0.51) P2RX7CYP2A13KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899296-B1 HISTAMINE-3 RECEPTOR ANTAGONISTS PFIZER PROD INC (US) 2010-11-17 EP claimed