SCHEMBL3379545

SCHEMBL3379545

Cc1cc(Nc2nc(NCCN)c(F)cc2C=O)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 8/20 0.40
ZAP70 P43403 7/20 0.38
CAMK1D Q8IU85 1/20 0.38
PRKCE Q02156 1/20 0.37
BTK Q06187 1/20 0.37
ITK Q08881 1/20 0.37
BCDIN3D Q7Z5W3 2/20 0.37
CDK1 P06493 2/20 0.36
PRKCA P17252 2/20 0.36
TAS2R14 Q9NYV8 1/20 0.36
RAPGEF4 Q8WZA2 2/20 0.36
SRC P12931 3/20 0.35
CDK2 P24941 1/20 0.35
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
KCNH2 Q12809 1/20 0.33
AURKB Q96GD4 1/20 0.33
IKBKB O14920 1/20 0.33
CDK11B P21127 1/20 0.33
CDK7 P50613 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14929435 0.83 SYK (0.56) SYKZAP70CAMK1DPRKCEBTK
SCHEMBL14911001 0.74 SYK (0.56) SYKZAP70CAMK1DPRKCEBTK
SCHEMBL14909820 0.72 SYK (0.65) SYKZAP70CAMK1DKCNH2AURKB
SCHEMBL14923850 0.67 SYK (0.71) SYKZAP70CAMK1DPRKCEBTK
SCHEMBL14929769 0.66 SYK (0.56) SYKZAP70KCNH2AURKB
SCHEMBL17018670 0.64 SYK (0.51) SYKZAP70CDK1KCNH2AURKB
SCHEMBL14923870 0.64 SYK (0.69) SYKZAP70CAMK1DPRKCEBTK
SCHEMBL14923793 0.64 SYK (0.65) SYKZAP70CAMK1DPRKCEBTK
SCHEMBL16559049 0.63 DHFR (0.38) SYKZAP70CAMK1DCDK1PRKCA
SCHEMBL13996789 0.62 TRPA1 (0.51) TAS2R14RAPGEF4NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012002577-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF 富士フイルム株式会社 (JP) 2012-01-05 WO disclosed