SCHEMBL3380116

SCHEMBL3380116

Cc1noc(C)c1OC(=O)N(C)CC1CC(Oc2cccc(CN3CCCC3)c2F)C1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 2/20 0.35
HRH3 Q9Y5N1 2/20 0.35
GRIN1 Q05586 3/20 0.34
GRIN2B Q13224 3/20 0.34
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 4/20 0.33
MEN1 O00255 3/20 0.33
P2RX7 Q99572 2/20 0.32
SIRT2 Q8IXJ6 3/20 0.32
TAS2R8 Q9NYW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3378689 0.91 HRH3 (0.39) CYP2D6ALDH1A1CYP3A4HRH3CYP2C9
SCHEMBL3380644 0.91 ALDH1A1 (0.39) CYP2D6ALDH1A1CYP3A4HRH3CYP2C9
Hydrochloric Acid SCHEMBL3380991 0.86 CYP2D6 (0.41) CYP2D6ALDH1A1CYP3A4HRH3GRIN1
Hydrochloric Acid SCHEMBL3380987 0.86 CYP2D6 (0.41) CYP2D6ALDH1A1CYP3A4HRH3GRIN1
SCHEMBL3375226 0.83 HRH3 (0.42) HRH3
SCHEMBL3381390 0.81 HTR2C (0.33) ALDH1A1HRH3KMT2AMEN1
SCHEMBL3377784 0.81 MEN1 (0.46) ALDH1A1HRH3GRIN1GRIN2BKMT2A
SCHEMBL3377782 0.81 MEN1 (0.46) ALDH1A1HRH3GRIN1GRIN2BKMT2A
SCHEMBL3377365 0.81 HRH3 (0.47) HRH3P2RX7
SCHEMBL3377536 0.80 KMT2A (0.38) ALDH1A1HRH3GRIN1GRIN2BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899296-B1 HISTAMINE-3 RECEPTOR ANTAGONISTS PFIZER PROD INC (US) 2010-11-17 EP claimed