SCHEMBL338191

SCHEMBL338191

CC1NC(=O)OC1c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 11/20 0.49
CA2 P00918 1/20 0.48
SLC6A2 P23975 1/20 0.46
ADRA1A P35348 1/20 0.46
HTR2B P41595 1/20 0.46
SLC6A3 Q01959 1/20 0.46
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4291 1.00 GRM5 (0.49) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL4687 1.00 GRM5 (0.49) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL3119262 1.00 GRM5 (0.49) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL8192290 1.00 GRM5 (0.49) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL5835621 1.00 GRM5 (0.49) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL5544656 1.00 GRM5 (0.49) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL8532996 1.00 GRM5 (0.49) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL6374631 1.00 GRM5 (0.49) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL27504027 0.98 GRM5 (0.48) GRM5CA2SLC6A2ADRA1AHTR2B
SCHEMBL5196221 0.91 GRM5 (0.57) GRM5CA2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 268 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030225161-A1 GABA and L-glutamic acid analogs for antiseizure treatment NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-12-04 US claimed
EP-0925292-B1 PROCESSES AND INTERMEDIATES FOR PREPARING SUBSTITUTED CHROMANOL DERIVATIVES PFIZER (US) 2003-09-10 EP claimed
US-6180238-B1 PARTICULARLY SUITABLE FOR USE IN INK JET PRINTING PROCESSES. XEROX CORPORATION 2001-01-30 US claimed
EP-0743574-B1 Migration imaging members XEROX CORP (US) 2000-12-27 EP claimed
EP-0743573-B1 Method for obtaining image contrast migration imaging members XEROX CORP (US) 2000-09-06 EP claimed
EP-0673784-B1 Recording sheets containing oxazole, isooxazole, oxazolidinone, oxazoline salts, morpholine, thiazole, thiazolidine, thiadiazole, and phenothiazine compounds XEROX CORP (US) 1999-10-27 EP claimed
US-5729266-A Recording sheets containing oxazole, isooxazole, oxazolidinone, oxazoline salt, morpholine, thiazole, thiazolidine, thiadiazole and phenothiazine compounds XEROX CORPORATION (US) 1998-03-17 US claimed
EP-0641330-A4 GABA AND L-GLUTAMIC ACID ANALOGS FOR ANTISEIZURE TREATMENT. UNIV NORTHWESTERN (US) 1997-05-28 EP claimed
EP-0672687-B1 Process for producing amino-functional cyclodextrin derivatives CONSORTIUM ELEKTROCHEM IND (DE) 1997-03-19 EP claimed
EP-0743574-A2 Migration imaging members XEROX CORPORATION (US) 1996-11-20 EP claimed
EP-0743573-A2 Method for obtaining image contrast migration imaging members XEROX CORPORATION (US) 1996-11-20 EP claimed
US-5563014-A SOFTENABLE LAYER CONTAINIG PHOTOSENSITIVE MARKING MATERIAL; TRANSPARENTIZING AGENT XEROX CORPORATION (US) 1996-10-08 US claimed
US-5536826-A OXAZOLIDINONE OR DERIVATIVE CONSORTIUM FUR ELEKTROCHEMISCHE INDUSTRIE GMBH (DE) 1996-07-16 US claimed
US-5514505-A SELECTIVE TRANSPARENTIZATION OF PHOTOSENSITIVE MIGRATION MARKING PARTICLES EMBEDDED NEAR THE SURFACE OF A SOFTENABLE LAYER SUPPORTED BY AN ELECTROCONDUCTIVE SUBSTRATE XEROX CORPORATION (US) 1996-05-07 US claimed
EP-0673784-A2 Recording sheets containing oxazole, isooxazole, oxazolidinone, oxazoline salts, morpholine, thiazole, thiazolidine, thiadiazole, and phenothiazine compounds XEROX CORPORATION (US) 1995-09-27 EP claimed
EP-0672687-A1 Process for producing amino-functional cyclodextrin derivatives Consortium für elektrochemische Industrie GmbH (DE) 1995-09-20 EP claimed
EP-0641330-A1 GABA AND L-GLUTAMIC ACID ANALOGS FOR ANTISEIZURE TREATMENT NORTHWESTERN UNIVERSITY (US) 1995-03-08 EP claimed
EP-0378657-B1 OXAZOLIDINONE PENETRATION ENHANCING COMPOUNDS RAJADHYAKSHA VITHAL J (US) 1994-02-02 EP claimed
WO-1993023383-A1 GABA AND L-GLUTAMIC ACID ANALOGS FOR ANTISEIZURE TREATMENT NORTHWESTERN UNIVERSITY (US) 1993-11-25 WO claimed
US-4960771-A TRANSDERMAL DELIVERY OF THERAPEUTIC AGENTS; DRUGS, SUNSCREENS, INSECT REPELLENTS, COSMETICS LVMH MOET HENNESSY LOUIS VUITTON, INC. 1990-10-02 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225161-A1 GABA and L-glutamic acid analogs for antiseizure treatment GABRB1, GABRE, GABRB2 GRM5 50/4885CA2 319/4885SLC6A2 1005/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.