SCHEMBL3383240

SCHEMBL3383240

CC(C)(C)c1ccnc(NC(=O)Cc2ccc(-c3cnc4cc(-c5ccccn5)ccn34)cc2F)c1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 18/20 0.49
KDR P35968 17/20 0.49
WNT3A P56704 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383022 0.93 FGFR3 (0.52) FGFR3KDR
SCHEMBL3382979 0.93 FGFR3 (0.48) FGFR3KDRWNT3A
SCHEMBL3178478 0.90 FGFR3 (0.52) FGFR3KDR
SCHEMBL3382504 0.88 KDR (0.47) FGFR3KDRWNT3A
SCHEMBL3385467 0.88 KDR (0.49) FGFR3KDRWNT3A
SCHEMBL3386163 0.88 WNT3A (0.42) FGFR3KDRWNT3A
SCHEMBL3381090 0.87 FGFR3 (0.49) FGFR3KDRWNT3A
SCHEMBL3189878 0.87 KDR (0.49) FGFR3KDR
SCHEMBL3385477 0.87 FGFR3 (0.41) FGFR3KDR
SCHEMBL3383517 0.86 KDR (0.44) FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed