SCHEMBL3383247

SCHEMBL3383247

Cc1cc(C(=O)Nc2ccc(-c3ccc4c(C(=O)O)n[nH]c4c3)cc2)c(C)o1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.53
AKR1C3 P42330 1/20 0.50
AKR1C2 P52895 1/20 0.50
AKR1C1 Q04828 1/20 0.50
NPC1 O15118 6/20 0.47
RAB9A P51151 5/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
LRRK2 Q5S007 1/20 0.46
MAPT P10636 3/20 0.45
ALDH1A1 P00352 3/20 0.45
PKM P14618 1/20 0.45
MAPK1 P28482 3/20 0.44
TP53 P04637 2/20 0.44
HSD11B1 P28845 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
FLT3 P36888 2/20 0.43
PRKAG1 P54619 1/20 0.42
PRKAA1 Q13131 1/20 0.42
PRKAB1 Q9Y478 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386328 0.87 HPGD (0.48) HPGDAKR1C3AKR1C2AKR1C1NPC1
SCHEMBL3386831 0.82 NPC1 (0.54) HPGDNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL3387486 0.80 DYRK1A (0.54) NPC1RAB9AMAPTALDH1A1FLT3
Hydrochloric Acid SCHEMBL3386776 0.79 DYRK1A (0.53) NPC1RAB9AMAPTALDH1A1FLT3
SCHEMBL3380466 0.76 PAK1 (0.47) ALDH1A1PRKAG1PRKAA1PRKAB1JAK2
SCHEMBL3382225 0.75 PRKAG1 (0.56) HPGDNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL3384808 0.75 PRKAA1 (0.53) NPC1RAB9ASMN1; SMN2KDM4EFLT3
SCHEMBL3386038 0.74 DYRK1A (0.48) FLT3PRKAG1PRKAA1PRKAB1JAK2
SCHEMBL3385551 0.74 SGK1 (0.47) NPC1RAB9ASMN1; SMN2MAPTMAPK1
SCHEMBL3385649 0.74 NPC1 (0.50) HPGDNPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010064875-A2 NOVEL INDAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS PROTEIN KINASE INHIBITORS FOR PROLIFERATIVE DISEASES TREATMENT, AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2010-06-10 WO claimed
WO-2010064875-A2 NOVEL INDAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS PROTEIN KINASE INHIBITORS FOR PROLIFERATIVE DISEASES TREATMENT, AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2010-06-10 WO disclosed