SCHEMBL3385649

SCHEMBL3385649

O=C(Nc1ccc(-c2ccc3c(C(=O)O)n[nH]c3c2)cc1)c1cnccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 14/20 0.50
RAB9A P51151 14/20 0.50
SMN1; SMN2 Q16637 7/20 0.50
KMT2A Q03164 2/20 0.49
DYRK1A Q13627 3/20 0.47
CLK2 P49760 1/20 0.47
CLK3 P49761 1/20 0.47
TP53 P04637 4/20 0.46
MAPT P10636 4/20 0.46
USP2 O75604 2/20 0.46
MEN1 O00255 1/20 0.46
POLB P06746 1/20 0.46
P2RY14 Q15391 1/20 0.46
ALDH1A1 P00352 2/20 0.45
TSHR P16473 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HTT P42858 1/20 0.45
HPGD P15428 1/20 0.45
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387266 0.85 RAB9A (0.60) NPC1RAB9ASMN1; SMN2KMT2ADYRK1A
SCHEMBL3380466 0.83 PAK1 (0.47) KMT2ADYRK1ACLK2CLK3POLB
SCHEMBL3386126 0.83 PTGDR2 (0.43) DYRK1AWNT1
SCHEMBL3383259 0.81 MAPT (0.57) SMN1; SMN2KMT2AMAPTMEN1ALDH1A1
SCHEMBL3386038 0.80 DYRK1A (0.48) DYRK1ACLK2CLK3WNT1
SCHEMBL3386831 0.79 NPC1 (0.54) NPC1RAB9ASMN1; SMN2TP53MAPT
SCHEMBL3386591 0.75 KDR (0.50) NPC1RAB9ASMN1; SMN2KMT2ADYRK1A
SCHEMBL3385551 0.74 SGK1 (0.47) NPC1RAB9ASMN1; SMN2KMT2ADYRK1A
SCHEMBL3383247 0.74 HPGD (0.53) NPC1RAB9ASMN1; SMN2KMT2ATP53
SCHEMBL3387655 0.73 PAK1 (0.53) DYRK1AWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010064875-A2 NOVEL INDAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS PROTEIN KINASE INHIBITORS FOR PROLIFERATIVE DISEASES TREATMENT, AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2010-06-10 WO claimed
WO-2010064875-A2 NOVEL INDAZOLE DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS PROTEIN KINASE INHIBITORS FOR PROLIFERATIVE DISEASES TREATMENT, AND A PHARMACEUTICAL COMPOSITION CONTAINING THE SAME AS AN ACTIVE INGREDIENT KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2010-06-10 WO disclosed