SCHEMBL3383608

SCHEMBL3383608

CC(Cc1cc(-c2ccn3c(-c4ccc(CC(=O)Nc5ncc(C6(O)CCC6)s5)c(F)c4)cnc3c2)ccn1)N1CCOCC1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
FGFR3 P22607 11/20 0.33
KDR P35968 9/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
PDGFRA P16234 1/20 0.32
SIK1 P57059 4/20 0.32
SIK2 Q9H0K1 4/20 0.32
SIK3 Q9Y2K2 4/20 0.32
CTSC P53634 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3380785 0.91 FGFR3 (0.36) SMN1; SMN2FGFR3KDR
SCHEMBL3384486 0.88 CCNE1 (0.37) SMN1; SMN2FGFR3KDRPDGFRASIK1
SCHEMBL3196988 0.88 FGFR3 (0.35) FGFR3KDRPSEN1PSEN2APH1B
SCHEMBL3196972 0.88 FGFR3 (0.35) FGFR3KDRPSEN1PSEN2APH1B
SCHEMBL3186881 0.88 FGFR3 (0.33) FGFR3KDRPDGFRASIK1SIK2
SCHEMBL3186871 0.88 FGFR3 (0.33) FGFR3KDRPDGFRASIK1SIK2
SCHEMBL3382693 0.85 WNT3A (0.41) SMN1; SMN2FGFR3KDR
SCHEMBL3379579 0.84 KDR (0.43) SMN1; SMN2FGFR3KDR
SCHEMBL3383109 0.84 KDR (0.35) FGFR3KDRCTSC
SCHEMBL13002537 0.83 KDR (0.34) FGFR3KDRCTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed