SCHEMBL3384206

SCHEMBL3384206

O=C(Cc1ccc(-c2cnc3cc(-c4ccccn4)ccn23)cc1F)Nc1ncc(C2(O)CCC2)s1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 18/20 0.45
FGFR3 P22607 17/20 0.45
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3379579 0.89 KDR (0.43) KDRFGFR3SMN1; SMN2
SCHEMBL3382693 0.87 WNT3A (0.41) KDRFGFR3SMN1; SMN2
SCHEMBL3385390 0.84 KDR (0.49) KDRFGFR3
SCHEMBL3385528 0.84 FGFR3 (0.46) KDRFGFR3MEN1RAB9AKMT2A
SCHEMBL3383557 0.83 KDR (0.44) KDRFGFR3
SCHEMBL3380785 0.82 FGFR3 (0.36) KDRFGFR3SMN1; SMN2
SCHEMBL4973341 0.82 FGFR3 (0.42) KDRFGFR3MEN1RAB9AKMT2A
SCHEMBL3187730 0.81 KDR (0.41) KDRFGFR3MEN1RAB9AKMT2A
SCHEMBL3381798 0.81 KDR (0.48) KDRFGFR3
SCHEMBL3383608 0.80 SMN1; SMN2 (0.34) KDRFGFR3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed