SCHEMBL3385159

SCHEMBL3385159

Cc1cc(-c2ccn3c(-c4ccc(NC(=O)N(OS(C)(=O)=O)c5cc(C(C)(C)C)on5)c(F)c4)cnc3c2)ccn1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 13/20 0.34
KDR P35968 13/20 0.34
PIK3CA P42336 2/20 0.34
MTOR P42345 2/20 0.34
MAPK13 O15264 1/20 0.34
MAPK14 Q16539 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
FLT3 P36888 1/20 0.33
PDGFRA P16234 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3381856 0.90 PIK3CA (0.45) FGFR3KDRPIK3CAMTORFLT3
SCHEMBL3385155 0.84 NPC1 (0.49) MAPK13MAPK14NPC1RAB9AFLT3
SCHEMBL3385688 0.79 PIK3CA (0.46) FGFR3KDRPIK3CAMTORFLT3
SCHEMBL3381118 0.74 NPC1 (0.54) FGFR3KDRMAPK13MAPK14NPC1
SCHEMBL3383303 0.74 NPC1 (0.52) KDRMAPK13MAPK14NPC1RAB9A
SCHEMBL3385839 0.73 NPC1 (0.51) KDRMAPK13MAPK14NPC1RAB9A
SCHEMBL3381854 0.73 NPC1 (0.49) FGFR3KDRPIK3CAMTORMAPK13
SCHEMBL3383068 0.73 NPC1 (0.50) FGFR3KDRMAPK13MAPK14NPC1
SCHEMBL3381837 0.73 NPC1 (0.48) MAPK13MAPK14NPC1RAB9AFLT3
SCHEMBL3383147 0.72 FGFR3 (0.40) FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed