SCHEMBL3385968

SCHEMBL3385968

CS(=O)(=O)c1ccc(-c2ccn3c(-c4ccc(NC(=O)Nc5cccc(C(F)(F)F)c5)c(F)c4)cnc3c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 14/20 0.53
KDR P35968 15/20 0.53
FLT3 P36888 2/20 0.48
NTRK1 P04629 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3386132 0.90 KDR (0.55) FGFR3KDRFLT3NTRK1
SCHEMBL3187562 0.84 KDR (0.56) FGFR3KDR
SCHEMBL3383213 0.83 RET (0.55) FGFR3KDRFLT3
SCHEMBL27686821 0.81 KDR (0.56) FGFR3KDR
SCHEMBL3195685 0.81 KDR (0.54) FGFR3KDRFLT3
SCHEMBL3186124 0.81 MGLL (0.49) FGFR3KDRFLT3NTRK1
SCHEMBL3320104 0.80 FGFR3 (0.79) FGFR3KDR
SCHEMBL3383303 0.80 NPC1 (0.52) KDRFLT3NTRK1
SCHEMBL3385985 0.79 EPHX2 (0.51) FGFR3KDR
SCHEMBL3190830 0.78 KDR (0.66) FGFR3KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128461-B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI 2010-12-22 CN disclosed
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed
CN-101128461-A Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI (US) 2008-02-20 CN disclosed