SCHEMBL338619

SCHEMBL338619

O=S(=O)(O)c1cc(S(=O)(=O)O)c2[nH]cnc2c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP1A2 P05177 1/20 0.36
LCK P06239 1/20 0.32
FYN P06241 1/20 0.32
ING2 Q9H160 1/20 0.32
FEN1 P39748 1/20 0.31
ALDH1A1 P00352 2/20 0.31
PARP1 P09874 1/20 0.30
CYP2C9 P11712 1/20 0.30
CASP6 P55212 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29636996 0.87 DUSP5 (0.33) CYP2C19HSD17B10CYP1A2FEN1KDM4E
SCHEMBL4749862 0.75 PARP1 (0.39) CYP2C19HSD17B10CYP1A2FEN1ALDH1A1
SCHEMBL28263803 0.75 DUSP5 (0.39) FEN1
SCHEMBL94274 0.72 PNP (0.38) CYP2C19HSD17B10LCKFYNING2
SCHEMBL10423950 0.72 LCK (0.36) CYP2C19HSD17B10LCKFYNING2
SCHEMBL29687182 0.72 PNP (0.38) CYP2C19HSD17B10LCKFYNING2
SCHEMBL2443793 0.71 LCK (0.32) LCKFYNING2
SCHEMBL28122236 0.71 PNP (0.37) LCKFYNING2FEN1ALDH1A1
SCHEMBL27613262 0.71 PNP (0.37) LCKFYNING2FEN1ALDH1A1
SCHEMBL571363 0.70 PRKCI (0.42) HSD17B10ALDH1A1CASP6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 104 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102448429-B Benzylidene malonates 巴斯夫欧洲公司 2018-03-06 CN claimed
EP-3052202-A1 SKIN TANNING EXTRACT DSM IP Assets B.V. (NL) 2016-08-10 EP claimed
WO-2015049366-A1 SKIN TANNING EXTRACT DSM IP ASSETS B.V. (NL) 2015-04-09 WO claimed
WO-2012116990-A2 NOVEL USE DSM IP ASSETS B.V. (NL) 2012-09-07 WO claimed
EP-2410974-A2 SUNSCREEN COMPOSITION COMPRISING HYDROXYAPATITE AS PHYSICAL SOLAR FILTER Kalichem Italia S.r.l. (IT) 2012-02-01 EP claimed
WO-2010109400-A2 SUNSCREEN PRODUCT COMPRISING HYDROXYAPATITE AS PHYSICAL FILTER KALICHEM ITALIA S.R.L. (IT) 2010-09-30 WO claimed
EP-4262727-A1 SELF-TANNING COMPOSITIONS DSM IP Assets B.V. (NL) 2023-10-25 EP disclosed
US-20220323334-A1 LIGHT AESTHETIC SUNSCREEN COMPOSITIONS JOHNSON & JOHNSON CONSUMER INC. 2022-10-13 US disclosed
WO-2022129265-A1 SELF-TANNING COMPOSITIONS DSM IP ASSETS B.V. (NL) 2022-06-23 WO disclosed
WO-2021142244-A1 SKIN TREATMENT METHODS AND COMPOSITIONS FOR TRANSDERMAL DELIVERY OF ACTIVE AGENTS TOPIX PHARMACEUTICALS, INC. (US) 2021-07-15 WO disclosed
EP-3817712-A1 AN ANTIMICROBIAL COMBINATION COMPOSITION COMPRISING GLYCEROL DERIVATIVES AND BICYCLIC COMPOUNDS Clariant International Ltd (CH) 2021-05-12 EP disclosed
EP-3802494-A1 PROCESS FOR FORMING 2-HYDROXYPYRIDINE-1-OXIDE OR DERIVATIVES THEREOF Clariant International Ltd (CH) 2021-04-14 EP disclosed
EP-3704134-A1 ANTIMICROBIAL TETRAPEPTIDES DSM IP Assets B.V. (NL) 2020-09-09 EP disclosed
US-6440401-B1 2-PHENYLBENZIMIDAZOLEDI- AND TRISULFONIC ACIDS; COSMETIC FORMULATIONS MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2002-08-27 US disclosed
US-4904564-A PHENOLIC-FORMALDEHYDE NOVOLAK; DIAZO SENSITIZER; IMIDAZOLE, BENZIMIDAZOLE, TRIAZOLE OR INDAZOLE TO INCREASE SOLUBILITY INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 1990-02-27 US disclosed
EP-0346650-A2 Process for imaging multi-layer resist structure International Business Machines Corporation (US) 1989-12-20 EP disclosed
EP-0139090-B1 PROCESS FOR THE PRE-TREATMENT OF POLYIMIDES SCHERING AKTIENGESELLSCHAFT (DE) 1988-07-27 EP disclosed
US-4517254-A ALKALI METAL HYDROXIDE, AMINOALKYLPOLYACID COMPOUNT SCHERING AKTIENGESELLSCHAFT (DE) 1985-05-14 US disclosed
EP-0139090-A1 Process for the pre-treatment of polyimides SCHERING AKTIENGESELLSCHAFT (DE) 1985-05-02 EP disclosed
US-4248632-A ACTIVATION OF A POLYMER SURFACE WITH A PALLADIUM COMPLEX SALT SCHERING AKTIENGESELLSCHAFT (DE) 1981-02-03 US disclosed