SCHEMBL3386743

SCHEMBL3386743

CC(C)N1CCN(C(=O)c2ccc3[nH]ccc3c2)CC1.CC(C)N1CCN(C(=O)c2ccc3c(ccn3CCN(C)C)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.48
DRD3 P35462 2/20 0.48
MAPK14 Q16539 1/20 0.46
HRH3 Q9Y5N1 5/20 0.44
CHRM2 P08172 1/20 0.42
OXTR P30559 2/20 0.42
GPR183 P32249 1/20 0.42
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
FASN P49327 1/20 0.41
SLC6A4 P31645 1/20 0.41
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3391353 0.95 PDK1 (0.47) DRD2DRD3MAPK14HRH3CHRM2
SCHEMBL3391336 0.91 HRH3 (0.53) HRH3OXTRSLC6A4
SCHEMBL3388425 0.87 HRH3 (0.52) DRD2DRD3MAPK14HRH3CHRM2
SCHEMBL3388732 0.86 MAPK14 (0.44) DRD2DRD3MAPK14HRH3CHRM2
SCHEMBL3387478 0.85 HRH3 (0.51) HRH3OXTRSLC6A4
SCHEMBL2219560 0.82 MAPK14 (0.60) DRD2DRD3MAPK14HRH3CHRM2
SCHEMBL3387643 0.78 HRH3 (0.51) HRH3OXTRSLC6A4
SCHEMBL3388360 0.78 HRH3 (0.43) DRD2DRD3MAPK14HRH3CHRM2
SCHEMBL3387941 0.76 MAPK14 (0.53) DRD2DRD3MAPK14HRH3CHRM2
SCHEMBL3388080 0.76 HRH3 (0.56) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029534-B1 1H-INDOL-5-YL-PIPERAZIN-1-YL-METHANONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-12-22 EP disclosed