SCHEMBL3387941

SCHEMBL3387941

CC(C)N1CCN(C(=O)c2ccc3[nH]ccc3c2)CC1.CC(C)N1CCN(C(=O)c2ccc3c(ccn3C[C@@H]3CCCN3Cc3ccccc3)c2)CC1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.53
OXTR P30559 3/20 0.42
CHRM2 P08172 1/20 0.42
ACHE P22303 2/20 0.41
HTR4 Q13639 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
HRH3 Q9Y5N1 3/20 0.40
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
MGLL Q99685 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CCR3 P51677 1/20 0.39
GHSR Q92847 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387892 0.92 OXTR (0.47) OXTRACHEHRH3KDM4E
SCHEMBL3386876 0.89 MAPK14 (0.54) MAPK14OXTRCHRM2ACHEHTR4
SCHEMBL3390449 0.81 MAPK14 (0.57) MAPK14OXTRCHRM2ACHEHTR4
SCHEMBL3383896 0.80 OXTR (0.48) OXTRACHEHRH3MGLLKDM4E
SCHEMBL3388360 0.80 HRH3 (0.43) MAPK14CHRM2ACHEHTR4HRH3
SCHEMBL3390881 0.79 MAPK14 (0.59) MAPK14OXTRCHRM2ACHEHTR4
SCHEMBL3390069 0.78 HRH3 (0.50) MAPK14OXTRACHEHRH3KDM4E
SCHEMBL3385999 0.78 HTR6 (0.52) OXTRHRH3
SCHEMBL3388425 0.77 HRH3 (0.52) MAPK14CHRM2HRH3DRD2DRD3
SCHEMBL3386743 0.76 DRD2 (0.48) MAPK14OXTRCHRM2HRH3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029534-B1 1H-INDOL-5-YL-PIPERAZIN-1-YL-METHANONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2010-12-22 EP disclosed