SCHEMBL3387185

SCHEMBL3387185

COc1ccc(CN2C(=O)NC3(CCN(CC4CN(CC5CCCCC5)CC4c4ccccc4)CC3)C2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.56
CCR5 P51681 17/20 0.51
OPRM1 P35372 1/20 0.45
OPRK1 P41145 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387190 1.00 OPRL1 (0.56) OPRL1CCR5OPRM1OPRK1MEN1
Hydrochloric Acid SCHEMBL3391698 0.99 OPRL1 (0.55) OPRL1CCR5OPRM1OPRK1MEN1
Hydrochloric Acid SCHEMBL3391692 0.99 OPRL1 (0.55) OPRL1CCR5OPRM1OPRK1MEN1
SCHEMBL3391696 0.88 CCR5 (0.50) OPRL1CCR5OPRM1OPRK1KMT2A
SCHEMBL3391693 0.88 CCR5 (0.50) OPRL1CCR5OPRM1OPRK1KMT2A
Hydrochloric Acid SCHEMBL3390786 0.87 CCR5 (0.49) OPRL1CCR5OPRM1OPRK1KMT2A
Hydrochloric Acid SCHEMBL3390783 0.87 CCR5 (0.49) OPRL1CCR5OPRM1OPRK1KMT2A
SCHEMBL3394539 0.83 CCR5 (0.44) OPRL1CCR5
SCHEMBL3394536 0.83 CCR5 (0.44) OPRL1CCR5
SCHEMBL3394174 0.83 CCR5 (0.49) OPRL1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7709642-B2 Spirohydantoin compounds and methods for the modulation of chemokine receptor activity VIROCHEM PHARMA, INC. (CA) 2010-05-04 US claimed