SCHEMBL3391553

SCHEMBL3391553

C#CCN(C)Cc1ccc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 15/20 0.61
POLQ O75417 4/20 0.51
LMNA P02545 2/20 0.41
USP2 O75604 1/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
ALDH1A1 P00352 1/20 0.41
BLM P54132 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393227 0.81 PYCR1 (0.63) PYCR1LMNAUSP2CYP3A4TSHR
SCHEMBL3394172 0.76 PYCR1 (1.00) PYCR1LMNAUSP2CYP3A4TSHR
SCHEMBL2324597 0.73 DAO (0.48) PYCR1POLQ
SCHEMBL25594632 0.70 CYP2C19 (0.64) POLQCYP3A4
SCHEMBL4416164 0.70 POLQ (0.51) POLQALDH1A1
SCHEMBL1538523 0.69 DAO (0.49) POLQ
SCHEMBL1993639 0.68 CES2 (0.52) POLQCYP3A4
SCHEMBL13349970 0.67 DAO (0.51) POLQ
SCHEMBL13644756 0.67 POLQ (0.46) POLQCYP3A4
SCHEMBL964552 0.67 DAO (0.46) POLQTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed