SCHEMBL3393227

SCHEMBL3393227

C#CCN(C)Cc1ccccc1C(F)(F)F

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 17/20 0.63
LMNA P02545 2/20 0.54
MAOA P21397 2/20 0.54
USP2 O75604 1/20 0.54
CYP3A4 P08684 1/20 0.54
TSHR P16473 1/20 0.54
MAOB P27338 1/20 0.54
ALDH1A1 P00352 1/20 0.53
BLM P54132 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3391553 0.81 PYCR1 (0.61) PYCR1LMNAMAOAUSP2CYP3A4
SCHEMBL12124971 0.81 SLC6A2 (0.54) ALDH1A1
SCHEMBL12831776 0.78 SLC6A4 (0.50) CYP3A4
SCHEMBL16269319 0.78 SCN8A (0.47) PYCR1LMNAMAOAUSP2CYP3A4
SCHEMBL18137967 0.78 SLC6A2 (0.56) ALDH1A1
SCHEMBL11473731 0.78 CARM1 (0.53)
SCHEMBL3812562 0.77 PYCR1 (0.69) PYCR1LMNAMAOAUSP2CYP3A4
SCHEMBL13965863 0.75 SLC6A2 (0.50)
SCHEMBL13975853 0.75 SLC6A2 (0.58)
SCHEMBL22651953 0.74 SLC6A2 (0.48) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed