SCHEMBL3391719

SCHEMBL3391719

CS(=O)(=O)c1ccc(CN2C(=O)NC3(CCN(CC4CN(S(=O)(=O)c5ccccc5)CC4c4ccccc4)CC3)C2=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 9/20 0.53
KDM1A O60341 1/20 0.43
MAOB P27338 1/20 0.43
KMT2A Q03164 2/20 0.40
SLC6A9 P48067 1/20 0.36
USP2 O75604 3/20 0.36
CYP3A4 P08684 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HIF1A Q16665 1/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
DRD2 P14416 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
LMNA P02545 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3391721 1.00 CCR5 (0.53) CCR5KDM1AMAOBKMT2ASLC6A9
Hydrochloric Acid SCHEMBL3389663 0.99 CCR5 (0.52) CCR5KDM1AMAOBKMT2ASLC6A9
Hydrochloric Acid SCHEMBL3389664 0.99 CCR5 (0.52) CCR5KDM1AMAOBKMT2ASLC6A9
SCHEMBL3392304 0.90 CCR5 (0.52) CCR5KMT2AALDH1A1MEN1MAPK1
SCHEMBL3392307 0.90 CCR5 (0.52) CCR5KMT2AALDH1A1MEN1MAPK1
Hydrochloric Acid SCHEMBL3388619 0.90 CCR5 (0.51) CCR5KMT2AALDH1A1MEN1MAPK1
Hydrochloric Acid SCHEMBL3388624 0.90 CCR5 (0.51) CCR5KMT2AALDH1A1MEN1MAPK1
SCHEMBL3391408 0.85 CCR5 (0.46) CCR5KDM1AMAOBKMT2AALDH1A1
SCHEMBL3391406 0.85 CCR5 (0.46) CCR5KDM1AMAOBKMT2AALDH1A1
SCHEMBL3391693 0.85 CCR5 (0.50) CCR5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7709642-B2 Spirohydantoin compounds and methods for the modulation of chemokine receptor activity VIROCHEM PHARMA, INC. (CA) 2010-05-04 US claimed