SCHEMBL3392239

SCHEMBL3392239

OB(O)c1ccc(C2=CCN(Cc3ccc(OC(F)(F)F)cc3)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
PPARG P37231 2/20 0.41
PPARA Q07869 2/20 0.41
FFAR1 O14842 1/20 0.41
LMNA P02545 1/20 0.40
KCNH2 Q12809 1/20 0.40
TNF P01375 1/20 0.40
NOD2 Q9HC29 1/20 0.40
NOD1 Q9Y239 1/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
BACE1 P56817 1/20 0.39
LSS P48449 1/20 0.39
HTR1A P08908 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3392726 0.85 ALDH1A1 (0.50) ALDH1A1TSHRMAPK1MEN1KMT2A
SCHEMBL5535869 0.77 PPARG (0.48) ALDH1A1MEN1KMT2APPARGPPARA
SCHEMBL5547325 0.76 PPARG (0.42) ALDH1A1TSHRMAPK1MEN1KMT2A
SCHEMBL20582537 0.76 PPARG (0.45) ALDH1A1TSHRMEN1KMT2APPARG
SCHEMBL5542216 0.75 PPARG (0.47) ALDH1A1TSHRMEN1KMT2APPARG
SCHEMBL3397349 0.74 ALDH1A1 (0.52) ALDH1A1TSHRMEN1KMT2ALMNA
SCHEMBL14438052 0.74 PPARG (0.51) ALDH1A1TSHRMEN1KMT2APPARG
SCHEMBL13070096 0.74 ALDH1A1 (0.42) ALDH1A1TSHRMAPK1MEN1KMT2A
Hydrochloric Acid SCHEMBL3392212 0.73 ALDH1A1 (0.41) ALDH1A1TSHRMAPK1MEN1KMT2A
SCHEMBL5535410 0.72 SIGMAR1 (0.46) ALDH1A1MEN1KMT2APPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed
WO-2010081904-A1 4 ( 1H) -PYRIDINONE DERIVATIVES AND THEIR USE AS ANTIMALARIA AGENTS GLAXO GROUP LIMITED (GB) 2010-07-22 WO disclosed