SCHEMBL3392272

SCHEMBL3392272

Cc1cc(C#N)ccc1-c1ccnc(NCc2cc(-c3ccccn3)[nH]n2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.54
FFAR1 O14842 2/20 0.38
METAP2 P50579 1/20 0.37
METAP1 P53582 1/20 0.37
CDK4 P11802 1/20 0.36
CDK2 P24941 1/20 0.36
TGFBR1 P36897 1/20 0.36
MAPK14 Q16539 1/20 0.36
CDC7 O00311 1/20 0.36
IGF1R P08069 1/20 0.35
FGFR1 P11362 1/20 0.35
KDR P35968 1/20 0.35
LRRK2 Q5S007 1/20 0.35
EGLN2 Q96KS0 1/20 0.34
ABCB1 P08183 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
CHEK1 O14757 1/20 0.34
KIT P10721 1/20 0.34
CRHR1 P34998 1/20 0.33
PDE5A O76074 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13425809 0.90 KCNH2 (0.49) KCNH2CDK4CDK2MAPK14CDC7
SCHEMBL3392059 0.85 KCNH2 (0.74) KCNH2FFAR1TGFBR1ABCB1ABCG2
SCHEMBL13425820 0.81 KCNH2 (0.40) KCNH2CDK4CDK2MAPK14
SCHEMBL3392275 0.78 KCNH2 (0.46) KCNH2FFAR1METAP2METAP1TGFBR1
SCHEMBL13425764 0.78 KCNH2 (0.53) KCNH2CDK4CDK2CDC7KIT
SCHEMBL13426284 0.78 KCNH2 (0.59) KCNH2TGFBR1MAPK14LRRK2ABCB1
SCHEMBL3395596 0.77 KCNH2 (0.40) KCNH2FFAR1METAP2METAP1TGFBR1
SCHEMBL3393337 0.76 KCNH2 (0.58) KCNH2TGFBR1ABCB1ABCG2CHEK1
SCHEMBL13426043 0.76 KCNH2 (0.43) KCNH2CHEK1
SCHEMBL13425594 0.75 KCNH2 (0.38) KCNH2FFAR1METAP2METAP1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed