SCHEMBL3392969

SCHEMBL3392969

O=C(O)Cc1c(O)cc(O)cc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.45
CA12 O43570 3/20 0.45
CA1 P00915 3/20 0.45
CA7 P43166 3/20 0.45
CA9 Q16790 3/20 0.45
CA14 Q9ULX7 3/20 0.45
TSHR P16473 2/20 0.45
ALDH1A1 P00352 2/20 0.45
PTGS2 P35354 2/20 0.45
ALOX5 P09917 1/20 0.45
POLB P06746 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PTPN1 P18031 1/20 0.41
PTPN11 Q06124 1/20 0.41
LCK P06239 2/20 0.40
EGFR P00533 1/20 0.40
HSD17B10 Q99714 3/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20983221 0.85 POLB (0.52) CA2CA12CA1CA7CA9
SCHEMBL39025 0.80 CA12 (0.45) CA2CA12CA1CA7CA9
SCHEMBL39033 0.77 PTPN1 (0.54) CA2CA12CA1CA7CA9
SCHEMBL9064155 0.76 CA1 (0.41) CA2CA12CA1CA7CA9
SCHEMBL39761 0.76 CA12 (0.41) CA2CA12CA1CA7CA9
SCHEMBL39571 0.74 KAT8 (0.50) PTPN1PTPN11KDM4EHPGDCYP3A4
SCHEMBL22660353 0.74 CA12 (0.40) CA2CA12CA1CA7CA9
SCHEMBL14968363 0.72 TAAR1 (0.50) CA2CA12CA1CA7CA9
SCHEMBL29002747 0.72 KDM4E (0.56) CA2CA12CA1CA7CA9
SCHEMBL3886521 0.72 ALDH1A1 (0.54) CA2CA12CA1CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188306-B2 Heat shock protein 90 inhibitors UNIVERSITY OF KANSAS (US) 2012-05-29 US disclosed
US-20100099865-A1 HEAT SHOCK PROTEIN 90 INHIBITORS UNIVERSITY OF KANSAS (US) 2010-04-22 US disclosed
US-7605288-B2 Heat shock protein 90 inhibitors UNIVERSITY OF KANSAS (US) 2009-10-20 US disclosed
US-20070197787-A1 Heat shock protein 90 inhibitors UNIVERSITY OF KANSAS 2007-08-23 US disclosed
US-7208630-B2 Heat shock protein 90 inhibitors UNIVERSITY OF KANSAS (US) 2007-04-24 US disclosed
WO-2006047740-A2 HEAT SHOCK PROTEIN 90 INHIBITORS UNIVERSITY OF KANSAS (US) 2006-05-04 WO disclosed
US-20060089495-A1 Heat shock protein 90 inhibitors NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2006-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060089495-A1 Heat shock protein 90 inhibitors HSP90AB2P, HSP90AB1, HSP90AA1 CA2 4190/4885CA12 4772/4885CA1 4406/4885
US-20070197787-A1 Heat shock protein 90 inhibitors HSP90AB2P, HSP90AB1, HSP90AA1 CA2 4190/4885CA12 4772/4885CA1 4406/4885
US-20100099865-A1 HEAT SHOCK PROTEIN 90 INHIBITORS HSP90AB2P, HSPH1, HSP90AA1 CA2 4053/4885CA12 4694/4885CA1 4126/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.