SCHEMBL3393526

SCHEMBL3393526

COc1ccc(C=Cc2cccc(Br)c2)cc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 9/20 0.55
CYP1A1 P04798 3/20 0.50
CYP1A2 P05177 3/20 0.50
CYP1B1 Q16678 3/20 0.50
NQO2 P16083 1/20 0.50
PTGS1 P23219 1/20 0.49
NFE2L2 Q16236 1/20 0.49
TUBB1 Q9H4B7 4/20 0.46
RELA Q04206 1/20 0.46
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44
TUBA4A P68366 1/20 0.44
TUBB4B P68371 1/20 0.44
TUBB3 Q13509 1/20 0.44
TUBB2A Q13885 1/20 0.44
TUBB8 Q3ZCM7 1/20 0.44
TUBA3E Q6PEY2 1/20 0.44
TUBA1A Q71U36 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393529 0.82 HSD17B3 (0.41) APPNQO2PTGS1NFE2L2RELA
SCHEMBL3395891 0.81 TUBB1 (0.64) APPCYP1A1CYP1A2CYP1B1NQO2
SCHEMBL5491895 0.77 RELA (0.71) APPCYP1A1CYP1A2CYP1B1NQO2
SCHEMBL5491899 0.77 RELA (0.71) APPCYP1A1CYP1A2CYP1B1NQO2
SCHEMBL15938427 0.76 TYR (0.58) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL15938428 0.76 TYR (0.58) CYP1A1CYP1A2CYP1B1NFE2L2TUBB1
SCHEMBL3362009 0.76 NQO2 (0.72) CYP1A1CYP1A2CYP1B1NQO2PTGS1
SCHEMBL3360764 0.76 NQO2 (0.72) CYP1A1CYP1A2CYP1B1NQO2PTGS1
SCHEMBL858370 0.75 ALDH1A1 (0.51)
SCHEMBL30424732 0.75 ALDH1A1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed