SCHEMBL3394007

SCHEMBL3394007

COC(=O)c1ccc(NCc2cc(O)c3ccccc3c2O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 1.00
HKDC1 Q2TB90 1/20 0.62
CA1 P00915 5/20 0.60
CA2 P00918 5/20 0.60
EGFR P00533 3/20 0.51
NOX4 Q9NPH5 1/20 0.51
HIF1A Q16665 3/20 0.51
ALDH1A1 P00352 2/20 0.50
RAB9A P51151 2/20 0.50
NPC1 O15118 1/20 0.50
HPGD P15428 1/20 0.50
AGTR1 P30556 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HSP90AA1 P07900 2/20 0.49
CYP19A1 P11511 1/20 0.48
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25442713 0.82 HKDC1 (0.70) ALOX5HKDC1CA1CA2EGFR
SCHEMBL17912677 0.78 GPR84 (0.64) ALOX5HKDC1CA1CA2RAB9A
SCHEMBL3394005 0.77 ALOX5 (0.62) ALOX5EGFRNOX4HIF1AALDH1A1
SCHEMBL5794016 0.77 HKDC1 (1.00) ALOX5HKDC1CA1CA2EGFR
SCHEMBL17912639 0.75 HDAC6 (0.71) ALOX5HKDC1CA1CA2HIF1A
SCHEMBL18415526 0.74 CA1 (1.00) ALOX5CA1CA2HIF1AALDH1A1
SCHEMBL13830817 0.74 CA1 (0.62) ALOX5HKDC1CA1CA2EGFR
SCHEMBL498241 0.73 HKDC1 (0.73) ALOX5HKDC1CA1CA2EGFR
SCHEMBL6262049 0.72 CA1 (0.72) ALOX5HKDC1CA1CA2HIF1A
SCHEMBL13934091 0.72 CA1 (0.87) ALOX5HKDC1CA1CA2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010033906-A2 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-03-25 WO disclosed