SCHEMBL3394483

SCHEMBL3394483

Cc1[nH]c(C)c(-c2c[nH]c(-c3ccc(CN4CCC(C(F)(F)F)CC4)cc3)cc2=O)c(=O)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TNKS O95271 6/20 0.37
PARP1 P09874 3/20 0.37
GRM2 Q14416 1/20 0.34
JAK3 P52333 1/20 0.34
MGAT2 Q10469 1/20 0.34
DRD2 P14416 4/20 0.33
DRD4 P21917 4/20 0.33
DRD3 P35462 4/20 0.33
RORC P51449 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
CRBN Q96SW2 1/20 0.33
IKZF3 Q9UKT9 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
MAP3K11 Q16584 1/20 0.33
CHEK1 O14757 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3397317 0.85 HRH3 (0.41) TNKSPARP1JAK3MGAT2DRD2
SCHEMBL3396969 0.84 MAP3K11 (0.39) TNKSPARP1GRM2HRH3MAP3K11
Hydrochloric Acid SCHEMBL3396774 0.84 GRM2 (0.40) GRM2JAK3DRD2DRD4DRD3
SCHEMBL3394839 0.80 SPR (0.32) DRD2DRD3
SCHEMBL3394476 0.79 JAK3 (0.36) GRM2JAK3MGAT2DRD2DRD4
SCHEMBL4565035 0.78 TNKS (0.39) TNKSPARP1
Hydrochloric Acid SCHEMBL3394572 0.78 DRD3 (0.33) DRD2DRD3
SCHEMBL3392240 0.77 PRKAB2 (0.36) CHEK1
SCHEMBL4475367 0.77 ADORA2A (0.39)
SCHEMBL4478743 0.77 SLC2A1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP claimed
EP-2246329-A1 4(1H)-pyridinone derivatives and their use as antimalaria agents Glaxo Group Limited (GB) 2010-11-03 EP disclosed