SCHEMBL3395282

SCHEMBL3395282

[CH2]c1n[nH]c2cc(Cl)ccc12

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP2K4 P45985 3/20 0.49
TRPA1 O75762 2/20 0.46
GSK3B P49841 2/20 0.44
GPR84 Q9NQS5 1/20 0.43
NOS1 P29475 2/20 0.41
DYRK1A Q13627 2/20 0.41
DAO P14920 1/20 0.41
ALDH1A1 P00352 1/20 0.40
CHEK1 O14757 1/20 0.40
PARP1 P09874 1/20 0.39
FADS1 O60427 1/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 1/20 0.37
JAK2 O60674 1/20 0.37
F7 P08709 1/20 0.36
F3 P13726 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3593032 0.79 MAP2K4 (0.50) MAP2K4TRPA1GSK3BGPR84NOS1
SCHEMBL14738828 0.79 MAP2K4 (0.63) MAP2K4TRPA1GSK3BNOS1DYRK1A
SCHEMBL4502873 0.78 PDPK1 (0.60) MAP2K4TRPA1GSK3BCHEK1JAK2
SCHEMBL15529807 0.76 GSK3B (0.48) MAP2K4TRPA1GSK3BGPR84NOS1
SCHEMBL2955244 0.76 MAP2K4 (0.55) MAP2K4TRPA1GSK3BGPR84NOS1
SCHEMBL30548014 0.76 GSK3B (0.48) MAP2K4TRPA1GSK3BGPR84NOS1
SCHEMBL3155790 0.76 CHEK1 (0.50) MAP2K4TRPA1GSK3BNOS1DYRK1A
SCHEMBL1553907 0.76 MAP2K4 (0.47) MAP2K4TRPA1GSK3BGPR84NOS1
SCHEMBL31735799 0.76 MAP2K4 (0.47) MAP2K4TRPA1GSK3BGPR84NOS1
SCHEMBL1551001 0.72 MAP2K4 (0.48) MAP2K4TRPA1GSK3BDAOALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233493-A1 Macrolides Pfizer Products Inc. (US) 2010-09-29 EP disclosed