SCHEMBL3395772

SCHEMBL3395772

CC(C)(C)C1CN(CCc2cc3c(cn2)OCCO3)CCN1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 14/20 0.36
GAA P10253 2/20 0.35
HTT P42858 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
SLC2A1 P11166 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3205594 0.74 CHRM2 (0.41) KCNH2MAPT
SCHEMBL5656515 0.74 KCNH2 (0.44) KCNH2HTTSLC2A1
SCHEMBL3504744 0.71 KDM2B (0.30)
SCHEMBL5748093 0.70 ALDH1A1 (0.38) KCNH2HTTKDM4EALDH1A1LMNA
SCHEMBL5439117 0.69 PTGS1 (0.36) KCNH2GAAKDM4EALDH1A1LMNA
SCHEMBL2076961 0.69 MAPK1 (0.37) GAAHTTKDM4EALDH1A1LMNA
SCHEMBL15191890 0.69 KCNJ1 (0.49) KCNH2
SCHEMBL3009489 0.69 CYP2J2 (0.32) KCNH2LMNA
SCHEMBL21820340 0.68 P2RX7 (0.32)
SCHEMBL3572416 0.68 ALOX15 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136807-B1 PYRROLO (3, 2, 1-IJ) QUINOLINE-4-ONE DERIVATIVES FOR TREATING TUBERCULOSIS GLAXO GROUP LTD (GB) 2010-11-03 EP disclosed