SCHEMBL3395849

SCHEMBL3395849

Oc1ccc(C=Cc2ccc(F)c(Br)c2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.65
MTOR P42345 2/20 0.65
TRPA1 O75762 2/20 0.63
VCP P55072 1/20 0.53
NQO2 P16083 2/20 0.52
LCK P06239 1/20 0.52
MAOB P27338 6/20 0.50
MAOA P21397 5/20 0.50
APP P05067 4/20 0.50
CA12 O43570 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA3 P07451 2/20 0.50
CA4 P22748 2/20 0.50
CA6 P23280 2/20 0.50
CA5A P35218 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
CA13 Q8N1Q1 2/20 0.50
CA14 Q9ULX7 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28785073 0.82 NFE2L2 (0.64) NPC1MTORTRPA1NQO2LCK
SCHEMBL25202875 0.81 CTSL (0.65) MAOBMAOAMEN1CYP3A4MAPT
SCHEMBL30382939 0.81 CTSL (0.65) MAOBMAOAMEN1CYP3A4MAPT
SCHEMBL25218023 0.81 CTSL (0.65) MAOBMAOAMEN1CYP3A4MAPT
SCHEMBL30383863 0.81 CTSL (0.65) MAOBMAOAMEN1CYP3A4MAPT
SCHEMBL6374804 0.78 NPC1 (1.00) NPC1MTORTRPA1NQO2LCK
SCHEMBL15093091 0.78 NPC1 (1.00) NPC1MTORTRPA1NQO2LCK
SCHEMBL29819435 0.78 NPC1 (1.00) NPC1MTORTRPA1NQO2LCK
SCHEMBL15093090 0.78 NPC1 (1.00) NPC1MTORTRPA1NQO2LCK
SCHEMBL38650704 0.78 VCP (0.58) NPC1MTORTRPA1VCPMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed