SCHEMBL3396554

SCHEMBL3396554

COc1ccccc1N1CCN(CCCNc2ccc(N)c(N)c2)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 9/20 0.62
DRD2 P14416 8/20 0.62
HTR2A P28223 3/20 0.62
HTR7 P34969 3/20 0.62
HTR6 P50406 3/20 0.62
DRD3 P35462 4/20 0.59
ADRA1A P35348 3/20 0.59
MAPT P10636 2/20 0.59
CYP3A4 P08684 2/20 0.59
ADRA2A P08913 2/20 0.59
ADRA2B P18089 2/20 0.59
ADRA2C P18825 2/20 0.59
LMNA P02545 1/20 0.59
ADRB2 P07550 1/20 0.59
ADRB1 P08588 1/20 0.59
CYP2C9 P11712 1/20 0.59
TSHR P16473 1/20 0.59
MAPK1 P28482 1/20 0.59
SLC6A4 P31645 1/20 0.59
CYP2C19 P33261 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26880831 0.89 DRD2 (0.67) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL11679210 0.85 LMNA (0.66) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL11676934 0.84 HTR1A (0.68) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL11676714 0.84 HTR1A (0.64) HTR1ADRD2HTR2AHTR7HTR6
Hydrochloric Acid SCHEMBL11677902 0.83 SMN1; SMN2 (0.63) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL253679 0.81 DRD2 (0.67) HTR1ADRD2HTR7DRD3ADRA1A
SCHEMBL8131826 0.80 HTR1A (0.65) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL16633469 0.80 DRD2 (0.59) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL3411899 0.80 SLC6A2 (0.76) HTR1ADRD2DRD3ADRA1AMAPT
SCHEMBL8130173 0.80 DRD2 (0.71) HTR1ADRD2HTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003418-A2 FUNCTIONALLY SELECTIVE LIGANDS OF DOPAMINE D2 RECEPTORS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2012-01-05 WO disclosed