SCHEMBL3397553

SCHEMBL3397553

FC(F)(F)c1cccc(N2CCN(c3ccncn3)CC2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 5/20 0.54
ALDH1A1 P00352 4/20 0.54
SIGMAR1 Q99720 2/20 0.54
HTR3E A5X5Y0 1/20 0.54
HTR3B O95264 1/20 0.54
HTR1D P28221 1/20 0.54
HTR2C P28335 1/20 0.54
HTR3A P46098 1/20 0.54
HTR3D Q70Z44 1/20 0.54
HTR3C Q8WXA8 1/20 0.54
KDM4E B2RXH2 1/20 0.53
POLB P06746 1/20 0.53
MAPT P10636 4/20 0.52
THRB P10828 1/20 0.52
DHFR P00374 1/20 0.51
RPS6KB1 P23443 1/20 0.49
AKT1 P31749 1/20 0.49
TSHR P16473 3/20 0.49
NPSR1 Q6W5P4 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27803379 0.82 RPS6KB1 (0.46) ALDH1A1MAPTDHFRRPS6KB1AKT1
SCHEMBL28226906 0.81 ALDH1A1 (0.77) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL27506706 0.79 ALDH1A1 (0.60) PHGDHALDH1A1SIGMAR1HTR3EHTR3B
SCHEMBL27846243 0.77 ALDH1A1 (0.52) PHGDHALDH1A1SIGMAR1HTR3EHTR3B
SCHEMBL2494773 0.77 DHFR (0.59) PHGDHALDH1A1SIGMAR1HTR3EHTR3B
Hydrochloric Acid SCHEMBL27803375 0.76 MAPT (0.53) ALDH1A1KDM4EMAPTSMN1; SMN2GAA
SCHEMBL9767811 0.75
SCHEMBL7455896 0.75 SIGMAR1 (0.56) ALDH1A1SIGMAR1KDM4EPOLBMAPT
SCHEMBL12706910 0.74 ALDH1A1 (0.72) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D
SCHEMBL9310480 0.74 MAPT (0.58) ALDH1A1SIGMAR1HTR3EHTR3BHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245017-A2 NOVEL HETEROCYCLES Orchid Research Laboratories Limited (IN) 2010-11-03 EP claimed
WO-2009095773-A2 NOVEL HETEROCYCLES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2009-08-06 WO claimed
EP-1973884-A2 NOVEL HETEROCYCLES Orchid Research Laboratories Limited (IN) 2008-10-01 EP claimed
WO-2007083182-A2 NOVEL HETEROCYCLES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-07-26 WO claimed