SCHEMBL3398749

SCHEMBL3398749

[CH2]C(=O)CNc1cnc2ccccc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.56
NPC1 O15118 6/20 0.56
KDM4E B2RXH2 5/20 0.56
SMN1; SMN2 Q16637 4/20 0.56
ALDH1A1 P00352 3/20 0.56
LMNA P02545 2/20 0.56
HPGD P15428 2/20 0.56
HTT P42858 2/20 0.56
GFER P55789 1/20 0.56
HDAC6 Q9UBN7 4/20 0.55
KDR P35968 1/20 0.55
POLB P06746 2/20 0.53
TSHR P16473 1/20 0.53
HSD17B10 Q99714 1/20 0.53
HDAC3 O15379 3/20 0.53
HDAC4 P56524 3/20 0.53
HDAC1 Q13547 3/20 0.53
HDAC7 Q8WUI4 3/20 0.53
HDAC2 Q92769 3/20 0.53
HDAC10 Q969S8 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836629 0.86 KDR (0.60) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL3395422 0.81 NPC1 (0.61) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL27617535 0.80 KDR (0.68) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL27679373 0.78 HDAC6 (0.58) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL2641717 0.77 HDAC1 (0.81) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL14461305 0.76 HDAC1 (0.72) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL27599000 0.76 HDAC1 (0.67) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL12895711 0.76 RAB9A (0.59) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL27866684 0.76 NPC1 (0.80) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL14075128 0.75 RAB9A (0.55) RAB9ANPC1KDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015703-A2 NOVEL 6-O-SUBSTITUTED 15-MEMBERED 8A- AND 9A-LACTAMS GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. (HR) 2010-02-11 WO disclosed