SCHEMBL3395422

SCHEMBL3395422

[CH2]C(=O)CNc1ccc2ncccc2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 8/20 0.61
POLB P06746 2/20 0.61
MAPT P10636 2/20 0.61
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
HDAC6 Q9UBN7 3/20 0.56
PABPC1 P11940 1/20 0.55
ALDH1A1 P00352 3/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
TSHR P16473 1/20 0.52
HSD17B10 Q99714 1/20 0.52
RAB9A P51151 6/20 0.51
HDAC1 Q13547 2/20 0.49
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1193017 0.87 NPC1 (0.63) NPC1POLBMAPTMEN1KMT2A
SCHEMBL1193628 0.83 ALDH1A1 (0.60) NPC1POLBMAPTMEN1KMT2A
SCHEMBL3398749 0.81 RAB9A (0.56) NPC1POLBMAPTMEN1KMT2A
SCHEMBL27599138 0.80 NPC1 (0.77) NPC1POLBMAPTMEN1KMT2A
SCHEMBL1193623 0.80 ALOX5 (0.56) NPC1POLBMAPTMEN1KMT2A
SCHEMBL2639005 0.77 HDAC6 (0.69) NPC1POLBMAPTMEN1KMT2A
SCHEMBL29944526 0.77 NPC1 (0.77) NPC1POLBMAPTMEN1KMT2A
SCHEMBL5142389 0.77 NPC1 (0.77) NPC1POLBMAPTMEN1KMT2A
SCHEMBL8209526 0.77 NPC1 (0.48) NPC1POLBMAPTMEN1KMT2A
SCHEMBL27599014 0.77 NPC1 (0.70) NPC1POLBMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015703-A2 NOVEL 6-O-SUBSTITUTED 15-MEMBERED 8A- AND 9A-LACTAMS GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. (HR) 2010-02-11 WO disclosed